壹号娱乐APP

壹号娱乐APP | ENGLISH
刘君羊
浏览::  宣布时间::2022年03月18日

0ADAA874E3C87B5894DB387262F_8DCFC7EC_58A4

基本情形

刘君羊,,,男,,,中共党员。。壹号娱乐APP药学与食物工程学院副教授,,,硕士研究生导师。。

个人简介及研究偏向

主要从事活性(海洋)自然产品的全合成、、、结构修饰和构效关系研究,,,完成了包括甾体、、、萜类、、、大环内脂类、、、环肽类等凌驾18个活性自然产品的全合成。。历年来主持国家自然科学基金面上基金、、、青年基金,,,国家重点实验室开放课题项目、、、广东省教育厅学科重点提升项目,,,深圳市面上项目等9项。。现在在J. Am. Chem. Soc.、、、Chem、、、Green Syn. Catal.、、、Org. Lett.、、、Chinese J. Chem.、、、Org. Chem. Front.、、、Chem. Commun.、、、J. Org. Chem.、、、Nature Chemistry等国际刊物上揭晓研究论文38篇,,,其中以(配合)第一作者/(配合)通讯作者揭晓28篇,,,申请专利6项,,,授权2项。。现在是广东省药理学会海洋药物药理专业委员会委员,,,国自然科学基金、、、广东省基础与应用基础研究基金项目评审专家,,,广东省高条理人才评审专家,,,Chemical Science, RSC Advances, Marine Drugs等杂志审稿人。。

7ADD8848676D3A956037DA6F91C_677611D0_7775

联系方式

地点::广东省江门市蓬江区东成村22号壹号娱乐APP药学与食物工程学院

邮编::529020

e-mail::liujy@wyu.edu.cn

事情履历

2022.02至今 ,,,壹号娱乐APP,,,药学与食物工程学院,,,副教授,,,硕士生导师;;;

2017.12至2022.02,,,南方科技大学,,,高级研究学者、、、研究助理教授/研究副教授;;;2012.10至2017.11,,,北京大学、、、香港理工大学、、、南方科技大学,,,博士后/访学;;;

教育及学习履历

2006.09-2012.01 北京大学 博士

2001.09-2005.07 南昌大学 本科

科研项目

1. 国家自然科学基金,,,面上项目,,,2024.01-2027.12,,,主持;;;

2. 国家自然科学基金,,,青年基金项目,,,2017.01-2019.12,,,主持;;;

3. 广东省教育厅重点建设学科科研能力提升项目,,,2022.1-2024.12,,,主持;;;

4. 国家重点实验室,,,开放课题项目,,,2023.1-2024.12,,,主持;;;

5. 深圳市科创委,,,面上项目,,,2020.06-2023.6,,,主持;;;

揭晓学术论文

1. Liu, Junyang; Wu, Jianlei; Fan, Jian-Hong; Yan, Xin; Mei, Guangjian; Li, Chuang-Chuang, Asymmetric Total Synthesis of Cyclocitrinol. J. Am. Chem. Soc. 2018, 140, (16), 5365-5369.

2. Liu, Xin#; Liu, Junyang#; Wu, Jianlei; Huang, Guocheng; Liang, Rong; Chung, Lung Wa; Li, Chuang-Chuang*, Asymmetric Total Synthesis of Cerorubenic Acid-III. J. Am. Chem. Soc. 2019, 141, (7), 2872-2877.

3. Liu, Junyang#; Liu, Xin#; Wu, Jianlei; Li, Chuang-Chuang*, Total Synthesis of Natural Products Containing a Bridgehead Double Bond. Chem 2020, 6, (3), 579-615.

4. Chen, Louxi; Zhang, Chao-Han; Liu, Junyang*; Sun, Jianwei*; Li, Chuang-Chuang*, Asymmetric Synthesis of the Tetracyclic Core of Venezuelaene B. Org. Lett. 2025, 27, (14), 3517-3520.

5. Chen, Louxi; Zhang, Chao-Han; Liu, Junyang*; Li, Chuang-Chuang*, Asymmetric synthesis of venezuelaene's core with a trans-fused [5-5] ring system. Chem. Commun. 2025, 61, (58), 10823-10826.

6. Feng, Jiaxuan; Liu, Junyang*; Ye, Tao, Total Synthesis, Stereochemical Assignment, and Structural Revision of HA 23. Org. Lett. 2025, 27, (33), 9299-9303.

7. Peng, Wenquan#; Han, Feipeng#; Liu, Junyang#; Wang, Chenqi; Minami, Atsushi; Oikawa, Hideaki; Guo, Yian; Ye, Tao, Thermolides D and E: Total Synthesis and Stereochemical Revision. Org. Lett. 2025, 27, (30), 8183-8188.

8. Wang, Chenqi; Liu, Junyang*; Ye, Tao*, Synergy of prediction rule and total synthesis in solving the stereochemical puzzle of eucalactam B. Org. Chem. Front. 2025, 12, (1), 70-75.

9. Jiang, Yangyang; Liu, Junyang*; Ye, Tao*, Total synthesis and stereochemical assignment of cubensci acid. Org. Chem. Front. 2025, 12, 4525–4529

10. Long, Xiong-En; Xing, Hailiang; He, Yixin; Meng, Xuanli; Ma, Yanling; Liu, Chang; Cao, Xi; Nan, Huiru; Cheng, Min-Jing*; Yan, Jia-Lei*; Liu, Junyang*, Total synthesis and biological evaluation of Koshidacin B, TAN-1746, and Ac-TAN-1746. BMC Chemistry 2025, 19, 213.

11. Liu, Haoyang; Xing, Hailiang; Yu, Peilan; Wang, Yanjie; Yan, Jia-Lei; Liu, Junyang*; Wang, Min*, Base-Controlled Synthesis of Heteroatom-Embedded 9-Membered Cycloalkynes and 6-Membered Sultams through Copper-Catalyzed Cyclization. J. Org. Chem. 2025, 90, (2), 984-993.

12. Nan, Huiru; Long, Xiong-En; He, Jianfei; Xing, Hailiang; Cheng, Min-Jing; Peng, Jin-Bao; Ye, Tao*; Yan, Jia-Lei*; Liu, Junyang*, Total Synthesis of the Marine Cyclic Depsipeptide Lagunamide D. Mar. Drugs 2025, 23, (3), 99.

13. Gu, Chen-Chen; Long, Xiong-En; Chen, Xiuping; Liu, Junyang*; Li, Chuang-Chuang*, Recent Natural Product Total Syntheses Involving Cycloadditions of Allenes. Chin. J. Chem. 2025, 43, (9), 1059-1077.

14. Liu, Junyang; Chen, Kai; Guo, Yian; Chen, Ying; Ye, Tao*, Total Synthesis of Rhizopodin Enabled by a Late-Stage Oxazole Ring Formation Strategy. Org. Lett. 2024, 26, (41), 8928-8933.

15. Yan, Jia-Lei; Nan, Huiru; Fang, Xiaoyu; Long, Xiong-En; Jiang, Yu; Liu, Junyang*, The isolation, bioactivity, and synthesis of natural products from Litsea verticillate with anti-HIV activities. Front. Pharmacol. 2024, 15, 1477878.

16. Xiao, Yi#; Liu, Junyang#; Jiang, Yangyang; Guo, Yian; Ye, Tao*, Total Syntheses and Stereochemical Assignment of Acremolides A and B. Molecules 2024, 29, (15), 3599.

17. Hou, Bao-Long*; Liu, Junyang*; Qiao, Chuang*; Li, Chuang-Chuang*, Total synthesis of natural products containing bicyclo[n.2.2] ring systems. Tetrahedron Lett. 2024, 135, 154871.

18. He, Yujie; Chen, Jintao; Jiang, Yu; Fang, Xiaoyu; Liu, Junyang*; Yan, Jia-Lei*, N-Heterocyclic Carbene Catalyzed Reactions Involving Acetylenic Breslow and/or Acylazolium as Key Intermediates. Chem. Rec. 2024, 24, (12), e202400165.

19. Liu, Junyang#; Tang, Shoubin#; Yan, Jia-Lei; Ye, Tao*, Design and Synthesis of Novel Helix Mimetics Based on the Covalent H-Bond Replacement and Amide Surrogate. Molecules 2023, 28, (2), 780.

20. Liu, Junyang; Chen, Hang; Wang, Min; He, Wangjin; Yan, Jia-Lei*, Organocatalytic asymmetric synthesis of P-stereogenic molecules. Front. Chem. 2023, 11.

21. Hui, Chunngai#, *; Wang, Zhuo#; Xie, Yusheng*; Liu, Junyang*, Contemporary synthesis of bioactive cyclobutane natural products. Green Synth. Catal. 2023, 4, (1), 1-6.

22. Liu, Junyang*; Chen, Ying; Luesch, Hendrik; Ye, Tao*, Total Synthesis of des-Thiomethyllooekeyolide A. Org. Lett. 2022, 24, (40), 7260-7264.

23. Wu, Jianlei#; Liu, Junyang#, *; Fan, Jian-Hong; Xie, Zhi-Dong; Qin, Hukun; Li, Chuang-Chuang*, Evolution of Routes for Asymmetric Total Synthesis of Cyclocitrinol Enabled by Type II [5+2] Cycloaddition?. Chin. J. Chem. 2021, 39, (5), 1247-1254.

24. Liu, Xin#; Liu, Junyang#; Wu, Jianlei; Li, Chuang-Chuang*, Enantioselective Total Synthesis of Cerorubenic Acid-III via Type II [5+2] Cycloaddition Reaction. J. Org. Chem. 2021, 86, (16), 11125-11139.

25. Liu, Xin#; Liu, Junyang#; Zhao, Jing; Li, Shaoping; Li, Chuang-Chuang*, Toward the Total Synthesis of Eurifoloid A. Org. Lett. 2017, 19, (10), 2742-2745.

26. Liu, Junyang; Wang, Lei; Zhang, Juefei; Xu, Zhengshuang*; Ye, Tao*, The total synthesis and stereochemical assignment of scytonemin A. Chem. Commun. 2016, 52, (5), 1002-1005.

27. Song, Liankai#; Liu, Junyang#; Gui, Honggang; Hui, Chunngai; Zhou, Jingjing; Guo, Yian; Zhang, Pengpeng; Xu, Zhengshuang*; Ye, Tao*, Synthesis of the Macrocyclic Core of Rhizopodin. Chem. - Asian J. 2013, 8, (12), 2955-2959.

28. Liu, Junyang; Ma, Xiao; Liu, Yuqing; Wang, Zhuo; Kwong, Shuqin; Ren, Qi; Tang, Shoubin; Meng, Yi; Xu, Zhengshuang*; Ye, Tao*, Total Synthesis and Stereochemical Revision of Burkholdac A. Synlett 2012, 23, (05), 783-787.

申请及授权专利

1. 刘君羊,,,南慧茹,,,龙雄恩,,,邢海亮,,,何健飞,,,马艳玲,,,一种环肽 Lagunamide D 的制备要领,,,2024-12-30,,,中国,,,2024119701774。。

2. 刘君羊,,,龙雄恩,,,南慧茹,,,邢海亮,,,刘昊洋,,,一种四环肽中心体化合物及其制备要领和应用,,,2024-09-06,,,中国,,,202411250389.5。。

3. 刘君羊,,,刘昊洋,,,邢海亮,,,王敏,,,一种六元环磺酰胺类化合物的制备要领,,,2024-07-12,,,中国,,,202410937674(公开)。。

4. 刘君羊,,,景显彤,,,陈娄曦,,,李闯创,,,虎皮楠生物碱骨架的合成要领,,,2022-02-11,,,中国,,,CN116621868A(公开)。。

5. 刘君羊,,,南慧茹,,,龙雄恩,,,闫加磊,,,一种化合物及其合成要领与在肌动卵白稳固剂的合成要领中的应用,,,2023-12-04,,,中国,,,ZL202311645681.2(授权)。。

6. 刘君羊,,,吴建磊,,,范建红,,,李闯创,,,甾体化合物的制备要领,,,2018-03-13,,,中国,,,ZL201810205745.X(授权)。。


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