
»ù±¾ÇéÐÎ
Ê¢îȾý£¬Å®£¬ºþÄϳ£µÂÈË£¬Öй²µ³Ô±¡£¡£¡£ÏÖÈÎÒ¼ºÅÓéÀÖAPPҩѧÓëʳÎ﹤³ÌѧԺ¸±½ÌÊÚ¡¢¡¢Ë¶Ê¿Éúµ¼Ê¦£»£»½ÃÅ-ÀûÎïÆÖ¹«¹²ÎÀÉúÑо¿ËùËù³¤¡£¡£¡£
ÁªÏµ·½Ê½
µØµã£º£º£º¹ã¶«Ê¡½ÃÅÊÐÅî½Çø¶«³É´å22ºÅ Ò¼ºÅÓéÀÖAPPҩѧÓëʳÎ﹤³ÌѧԺ
Óʱࣺ£º£º529020
ÓÊÏ䣺£º£ºwyuchemszj@126.com
ÊÂÇéÂÄÀú
2015Äê5ÔÂÖÁ½ñ£¬Ò¼ºÅÓéÀÖAPP£¬Ò©Ñ§ÓëʳÎ﹤³ÌѧԺ£¬×¨ÈÎÎ÷ϯ
2017Äê1ÔÂÖÁ2017Äê3Ô£¬Ó¢¹úÀûÎïÆÖÈÈ´ø²¡Ñ§Ôº£¬»á¼ûѧÕß
2023Äê8ÔÂÖÁ2023Äê12Ô£¬Ó¢¹úÀûÎïÆÖÈÈ´ø²¡Ñ§Ôº£¬»á¼ûѧÕß
½ÌÓý¼°Ñ§Ï°ÂÄÀú
2004Äê9ÔÂÖÁ2008Äê6Ô£¬ÉÂÎ÷ʦ·¶´óѧ£¬Ñ§Ê¿
2006Äê9ÔÂÖÁ2007Äê6Ô£¬º«¹ú˳ÌìÏç´óѧ£¬½»Á÷Áôѧ
2008Äê9ÔÂÖÁ2014Äê12Ô£¬¹ã¶«¹¤Òµ´óѧ£¬²©Ê¿£¨Ë¶²©Á¬¶Á£©
2011Äê12ÔÂÖÁ2014Äê9Ô£¬·¨¹ú°ÍÀèµÚÆß´óѧ£¬²©Ê¿
Ö÷ÒªÑо¿Æ«Ïò
ÎÃó·µÈҽѧÀ¥³æµÄ»¯Ñ§·À¿Ø£¬×ÔÈ»²úÆ·×ÊÔ´¿ª·¢ÓëʹÓ㬹¦Ð§»¯×±Æ·µÄÑо¿Ó뿪·¢
½ÒÏþѧÊõÂÛÎÄ
1) Yuling Li, Jialun Zou, Xiaofei Ren, Wenjiao Li, Weifeng Wu, Qiwei Xuan, Hanwen Miao, Yajie Chen, Chi-Sing Lee, Zhaojun Sheng*. Discovery of ¦Á-hexyl cinnamaldehyde and its derivatives as novel larvicides against Aedes albopictus. Arabian Journal of Chemistry, 2024, 17 (9), 105873.£¨ÖпÆÔº¶þÇø£©
2) Xiaofei Ren, Wenjiao Li, Jingmiao Zhang, Yingxiang Zhu, Xiaohui Hou, Hanwen Miao, Ximing Xu, Dongjing Zhang*, and Zhaojun Sheng*. Screening of botanical spatial mosquito repellents from 64 essential oils and their interactions with odorant binding protein-3. Journal of Applied Entomology, 2024, published online. https://doi.org/10.1111/jen.13330£¨ÖпÆÔºÈýÇø£©
3) Yuling Li, Weifeng Wu, Rongchao Jian, Xiaofei Ren, Xiaole Chen, Weiqian David Hong, Min Wu, Jinglin Cai, Canyao Lao, Ximing Xu, Zhaojun Sheng*. Larvicidal, acetylcholinesterase inhibitory activities of four essential oils and their constituents against Aedes albopictus, and nanoemulsion preparation, Journal of Pest Science, 2023, 96: 961-971. £¨ÖпÆÔºÒ»Çø£©
4) Weifeng Wu, Yu Yang, Yingmiao Feng, Xiaofei Ren, Yuling Li, Wenjiao Li, Jietong Huang, Lingjia Kong, Xiaole Chen, Zhongze Lin, Xiaohui Hou, Longlai Zhang, Yajie Chen, Zhaojun Sheng*, Weiqian Hong*. Study of the repellent activity of 60 essential oils and their main constituents against Aedes albopictus, and nano-formulation development, Insects, 2022, 13, 1077. £¨ÖпÆÔº¶þÇø£©
5) Rongchao Jian, Yuan Lin, Yuling Li, Weifeng Wu, Xiaofei Ren, Zhanyuan Liang, Lingjia Kong, Jinglin Cai, Canyao Lao, Min Wu, Wenhua Chen, Jing Chen*, Weiqian David Hong*, Zhaojun Sheng*. Larvicidal activity of two Rutaceae plant essential oils and their constituents against Aedes albopictus (Diptera: Culicidae) in multiple formulations, Journal of Medical Entomology, 2022, 59(5): 1669-1677. £¨ÖпÆÔºÈýÇø£©
6) Panpan Wu, Hao He, Hang Ma, Borong Tu, Jiahao Li, Shengzhu Guo, Silin Chen, Nana Cao, Wende Zheng, Xiaowen Tang, Dongli Li, Xuetao Xu, Xi Zheng, Zhaojun Sheng*, Weiqian David Hong*, Kun Zhang*. Oleanolic acid indole derivatives as novel ¦Á-glucosidase inhibitors: Synthesis, biological evaluation, and mechanistic analysis, Bioorganic Chemistry, 2021, 107, 104580. £¨ÖпÆÔº¶þÇø£©
7) Zhaojun Sheng, Rongchao Jian, Fangying Xie, Bin Chen, Kun Zhang, Dongli Li, Wenhua Chen, Chiguang Huang, Yan Zhang, Litao Hu, Denggao Zhao, Xi Zheng, Panpan Wu*, Weiqian David Hong. Screening of larvicidal activity of 53 essential oils and their synergistic effect for the improvement of deltamethrin efficacy against Aedes albopictus, Industrial Crops and Products, 2020, 145, 112131. £¨ÖпÆÔºÒ»Çø£©
8) Xiaole Chen, Min Gao, Rongchao Jian, Weiqian David Hong, Xiaowen Tang, Yuling Li, Denggao Zhao, Kun Zhang, Wenhua Chen, Xi Zheng, Zhaojun Sheng*, Panpan Wu*. Design, synthesis and ¦Á-glucosidase inhibition study of novel embelin derivatives, Journal of Enzyme Inhibition and Medicinal Chemistry, 2020, 35(1), 565-573. £¨ÖпÆÔº¶þÇø£©
9) Zhaojun Sheng*?, Siyuan Ge?, Min Gao, Rongchao Jian, Xiaole Chen, Xuetao Xu, Dongli Li, Kun Zhang, Wen-Hua Chen*. Synthesis and biological activity of embelin and its derivatives: An overview, Mini-Reviews in Medicinal Chemistry, 2020, 20, 396-407. £¨ÖпÆÔºÈýÇø£©
10) Xuetao Xu, Jie Chen, Zhiqing Lin, Dongli Li, Kun Zhang, Zhaojun Sheng*, ShaohuaWang*, Shun Zhu, Abdullah M. Asiri. Synthesis and anti-inflammatory effects of oxaprozin-paeonol ester, Chinese Journal of Organic Chemistry, 2019, 39, 2958-2964. £¨ÖпÆÔºÈýÇø£©
11) Zhaojun Sheng, Yiming Shi, Ximing Xu, S¨¦bastien Bellynck, Kun Zhang, Zhiyun Du, Xuetao Xu, Fran?ois Maurel, Chang-Zhi Dong*. Development of XIAP antagonists on the basis of de novo 8,5-fused bicyclic lactam, ChemistryOpen, 2019, 8, 34-40. £¨ÖпÆÔºÈýÇø£©
12) Xiaole Chen, Chiguang Huang, Rongchao Jian, Yan Zhang, Weifeng Wu, Xiaowen Tang, Qiankai Tan, Zhaojun Sheng*, Kun Zhang*. Optimization of microwave-assisted extraction of soluble dietary fiber from potato pulp and its properties, Journal of Food Processing and Preservation, 2019, 43, e14204. £¨ÖпÆÔºËÄÇø£©
13) Zhaojun Sheng*, Siyuan Ge, Ximing Xu, Yan Zhang, Panpan Wu, Kun Zhang, Xuetao Xu, Chen Li, Denggao Zhao and Xiaowen Tang. Design, synthesis and evaluation of cinnamic acid ester derivatives as mushroom tyrosinase inhibitors, MedChemComm (ÏÖÃûRSC Medicinal Chemistry), 2018, 9, 853-861. £¨ÖпÆÔºÈýÇø£©
14) Zhaojun Sheng?*, Ruhan Ye?, Siyuan Ge, Chenggang Wang, Xuetao Xu, Guangwen Zhang and Ping Luo. A validated RP-HPLC method for quantitative determination of related impurities of cholic acid bulk drugs, Acta Chromatographica, 2018, 30(2), 114-118. £¨ÖпÆÔºËÄÇø£©
15) Zhaojun Sheng, Changzhi Dong*, Zhiyun Du, Yiming Shi, Frederique Pallois, Yang Lu, Kun Zhang*. Acid-induced atypical spontaneous conversion of 5-amino-2,6-dioxooctahydro-1H-pyrrolo[2,1-d][1,5]oxazocine into 4-(hydroxyl methyl)-2,5-dioxooctahydro-1H-pyrrolo[1,2-d][1,4]diazepine, Research on Chemical Intermediate, 2015, 41(10): 7179-7187. £¨ÖпÆÔºËÄÇø£©
ÊÚȨרÀû
1) Ê¢îȾý£¬ÀîîÚÁ壬Îâΰ·å£¬ÈÎС·É£¬ºéΪǫ. Ò»ÖÖºú½·À໯ºÏÎï¼°ÆäÖÆ±¸ÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2022 1 1043660.9£¬ÊÚȨͨ¸æÈÕ£º£º£º2024Äê8ÔÂ27ÈÕ¡£¡£¡£
2) Ê¢îȾý£¬ÀîîÚÁ壬Îâΰ·å£¬ºéΪǫ. Ò»ÖÖÈâ¹ðËáÑÜÉúÎïÔÚÎóæ·ÀÖÎÖеÄÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2022 1 1017248.X£¬ÊÚȨͨ¸æÈÕ£º£º£º2024Äê5ÔÂ14ÈÕ¡£¡£¡££¨ÒÑתÈã©
3) Ê¢îȾý£¬¸ßÃô£¬³ÂСÀÖ£¬¼òÈÙ³¬£¬ÌÆÐ¡ÎÄ£¬ºéΪǫ. Ò»ÖÖ»ùÓÚ¶ÔôÇ»ù±½õ«¹Ç¼Ü¦Á-ÆÏÌÑÌÇÜÕøÒÖÖÆ¼Á¼°ÆäÖÆ±¸ÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2019 1 0341315.5£¬ÊÚȨͨ¸æÈÕ£º£º£º2022-02-08.£¨ÒÑתÈã©
4) Ê¢îȾý£¬³ÂСÀÖ£¬¼òÈÙ³¬£¬ÌÆÐ¡ÎÄ£¬ÀîîÚÁ壬ÎâÅÎÅΣ¬ÕÅŸj. Ò»ÖÖº¬×ÔȻֲÎᆱÓÍÔöЧ¼ÁµÄɱÎÃ×éºÏÎï¼°ÆäÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2019 1 0980396.3£¬ÊÚȨͨ¸æÈÕ£º£º£º2021-04-30. £¨ÒÑתÈã©
5) Ê¢îȾý£¬¸ð˼æÂ£¬ÕÅÑ࣬ÕÅŸj. Ò»ÖÖ°ë×ÔȻȪԴµÄÀÒ°±ËáøÒÖÖÆ¼Á¼°ÆäÖÆ±¸ÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2017 1 1241832.2£¬ÊÚȨͨ¸æÈÕ£º£º£º2020-10-09. £¨ÒÑתÈã©
6) Ê¢îȾý£¬ÀîîÚÁ壬Îâΰ·å£¬ÈÎС·É£¬ºéΪǫ. Ò»ÖÖ¼ÐÐÄÐͶà±ÛÐÐΪ²â¶¨ÒÇ£¬ÉêÇëºÅ£º£º£ºZL 2022 2 2227435.2£¬ÊÚȨͨ¸æÈÕ£º£º£º2023Äê04ÔÂ25ÈÕ. £¨ÒÑתÈã©
7) Ê¢îȾý£¬Îâΰ·å£¬ºéΪǫ£¬ÀîîÚÁ壬¼òÈÙ³¬. Ò»ÖÖ³ÉÎÃιѪËÇÑø×°±¸£¬×¨ÀûºÅ£º£º£ºZL 2021 2 2055986.0£¬ÊÚȨͨ¸æÈÕ£º£º£º2022Äê2ÔÂ18ÈÕ. £¨ÒÑתÈã©
8) Ê¢îȾý£¬¼òÈÙ³¬£¬³ÂСÀÖ£¬¸ßÃô£¬ÎâÅÎÅΣ¬ºéΪǫ£¬»Æ³Ø¹â£¬ÀÀû. Ò»ÖÖ±ãЯʽµç¶¯ÎüÎÃÆ÷£¬×¨ÀûºÅ£º£º£ºZL 2019 2 0308180.8£¬ÊÚȨͨ¸æÈÕ£º£º£º2019-12-31.
9) ¶³¤ÖΣ¬Ê¢îȾý£¬ÕÅŸj£¬Ê·Ò»Ãù£¬¶ÅÖ¾ÔÆ. Ò»ÖÖÔÓ»¯¿¹°©Ò©Îï¼°ÆäÖÆ±¸ÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2016 1 0529964.4£¬ÊÚȨͨ¸æÈÕ£º£º£º2017-11-03.
10) ¶³¤ÖΣ¬Ê¢îȾý£¬ÕÅŸj£¬¶ÅÖ¾ÔÆ. Ò»ÖÖ·ÇëÄÀàµòÍöÒÖÖÆÂѰ×Þ׿¹¼Á¼°ÆäºÏ³ÉÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2016 1 0038275.3£¬ÊÚȨͨ¸æÈÕ2018-04-13.
11) ¶³¤ÖΣ¬Ê¢îȾý£¬ÕÅŸj£¬¶ÅÖ¾ÔÆ. Ò»ÖÖµòÍöÒÖÖÆÂѰ׵ÄÀàëÄÞ׿¹¼Á¼°ÆäºÏ³ÉÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2016 1 0036840.2£¬ÊÚȨͨ¸æÈÕ£º£º£º2019-09-20
12) ¶³¤ÖΣ¬Ê¢îȾý£¬ÕÅŸj£¬Ê·Ò»Ãù£¬¶ÅÖ¾ÔÆ. Ò»ÖÖ¶à°Ðµã¿¹°©Ò©Îï¼°ÆäÖÆ±¸ÒªÁìÓëÓ¦Óã¬×¨ÀûºÅ£º£º£ºZL 2016 1 0530047.8£¬ÊÚȨͨ¸æÈÕ£º£º£º2019-10-29
13) ÁÖÖÒÔó£¬ÕÅÇåÃñ£¬ÎâÅÎÅΣ¬Ê¢îȾý. Ò»ÖÖÂÁ̼ËáÃ¾Æ·Î¶Æ¬ÖÆ±¸ÓÃÖÆÁ£×°±¸¼°ÂÁ̼ËáþƷζƬÉú²ú¹¤ÒÕ£¬×¨ÀûºÅ£º£º£ºZL 2019 1 0388393.0£¬ÊÚȨͨ¸æÈÕ£º£º£º2020-04-07.
¿ÆÑÐÏîÄ¿£¨Ö÷³Ö£©£º£º£º
1) ÐÂÐÍàŵͪÉúÎïµç×ÓµÈÅÅÌåµÄÉè¼Æ¡¢¡¢ºÏ³É¼°Ò©´ú¶¯Á¦Ñ§Ñо¿£¬Ò¼ºÅÓéÀÖAPP¸Û°ÄÁªºÏÑз¢»ù½ð£¬2021WGALH10£¬2022Äê7ÔÂÖÁ2025Äê6Ô£¬Ö÷³Ö¡£¡£¡£
2) ÎÃ³æ¿ØÖÆÒ©¼ÁÑо¿ºÍ²úÆ·¿ª·¢£¬ÉîÛÚÊÐγÐſƼ¼ÓÐÏÞ¹«Ë¾Î¯ÍÐÏîÄ¿£¬HX23140£¬2023Äê8ÔÂ30ÈÕÖÁ2026Äê8ÔÂ30ÈÕ£¬Ö÷³Ö¡£¡£¡£
3) ÎÞ»¼×Ó¼Ó¹¤¹¤ÒÕÑо¿¼°²úÆ·¿ª·¢£¬ºþÄÏÎÞ»¼×ÓÅ©ÁÖ¿ªÕ¹ÓÐÏÞ¹«Ë¾Î¯ÍÐÏîÄ¿£¬HX23080£¬2023Äê6ÔÂÖÁ2025Äê5Ô£¬Ö÷³Ö¡£¡£¡£
4) ÐÂÐÍË®ÈÜÐÔÞô±´ËØÑÜÉúÎïµÄÉè¼Æ¡¢¡¢ºÏ³É¼°¿¹°©»îÐÔÑо¿£¬¹ã¶«Ê¡×ÔÈ»¿ÆÑ§»ù½ð£¬2016A030310441£¬2016Äê6ÔÂÖÁ2019Äê5Ô£¬Ö÷³Ö¡£¡£¡£
5) ΣÏÕ·ÏÎïÖ¸ÎÆÆÊÎöÒªÁìÑо¿¼°Ö¸ÎÆ¿ìËÙ¼ì²âÊÔ¼ÁºÐµÄÑÐÖÆ£¬¹ã¶«Ê¡¿Æ¼¼×¨Ïî×ʽ𣨡°´óרÏî+ʹÃüÇåµ¥¡±£©ÅàÓý׳´ó¿Æ¼¼ÌØÅÉÔ±²½¶ÓºÍ¿ÆÑÐÏàÖúÏîÄ¿£¬2023019£¬2023Äê06ÔÂ01ÈÕÖÁ2026Äê05ÔÂ31ÈÕ£¬Ö÷³Ö¡£¡£¡£
6) ¶÷ƽÂíÁåÊíÔüµÄ×ÛºÏʹÓü°Ó¦Óÿª·¢£¬¶÷ƽÊÐũҵ¾ÖίÍÐÏîÄ¿£¬HX16137£¬2017Äê6ÔÂÖÁ2019Äê5Ô£¬Ö÷³Ö¡£¡£¡£
7) ÏÖ´úÖÐÒ©ÖÊ¿ØÖ¸ÎÆÍ¼Æ×ÊÖÒÕµÄÓ¦Óûù´¡Ñо¿£¬ÌØÒ»Ò©ÒµÎ¯ÍÐÏîÄ¿£¬HX21072£¬2019Äê6ÔÂÖÁ2021Äê12Ô£¬Ö÷³Ö¡£¡£¡£
8) ¸ÊÓÍÁ×ËáÄÆµÄºÏ³É¹¤ÒÕÑо¿£¬Ì¨É½ÐÂÄþÖÆÒ©Î¯ÍÐÏîÄ¿£¬HX21169£¬2021Äê10ÔÂÖÁ2022Äê3Ô£¬Ö÷³Ö¡£¡£¡£
9) ½ðÊôÎÛÄà×ÊÔ´»¯ÏîÄ¿¼ì²âÊÖÒÕ¿ª·¢£¬½ÃÅвƲúÇéÐιܼÒÊÖÒÕÓÐÏÞ¹«Ë¾Î¯ÍÐÏîÄ¿£¬HX21122£¬2021Äê7ÔÂÖÁ2022Äê6Ô£¬Ö÷³Ö¡£¡£¡£
10) Þô±´ËØÑÜÉúÎïÀàµòÍöÒÖÖÆÂѰ×Þ׿¹¼ÁµÄºÏ³É¼°¹¹Ð§¹ØÏµÑо¿£¬Ò¼ºÅÓéÀÖAPPÇàÄê¿ÆÑлù½ð£¬2015zk03£¬2015Äê11ÔÂÖÁ2018Äê10Ô£¬Ö÷³Ö¡£¡£¡£
11) ¸ÌÆÕ²èµÄ»¯Ñ§ÒòËØÆÊÎö¼°½µÑªÌǹ¦Ð§Ñо¿£¬Ò¼ºÅÓéÀÖAPP²©Ê¿¿ÆÑÐÆô¶¯ÏîÄ¿£¬2016BS18£¬2015Äê10ÔÂÖÁ2018Äê9Ô£¬Ö÷³Ö¡£¡£¡£
12) ×ÔȻֲÎᆱÓÍÓëºÏ³É¿¹ÎÃÒ©ÐͬЧӦÓë×÷ÓûúÀíÑо¿£¬½ÃÅÊлù´¡ÓëÀíÂÛ¿ÆÑ§Ñо¿Àà¿Æ¼¼ÍýÏëÏîÄ¿£¬2019030102100008866£¬2019Äê5ÔÂÖÁ2021Äê4Ô£¬Ö÷³Ö¡£¡£¡£
13) ÐÂÐÍÄâ³ý³æ¾Õõ¥ÀàÒ©ÎïµÄÉè¼Æ¡¢¡¢ºÏ³É¼°¿¹ÎûîÐÔÆÀ¼Û£¬½ÃÅÊлù´¡ÓëÀíÂÛ¿ÆÑ§Ñо¿Àà¿Æ¼¼ÍýÏëÏîÄ¿£¬2021030101400004873£¬2021Äê6ÔÂÖÁ2023Äê6Ô£¬Ö÷³Ö¡£¡£¡£
»ñ½±£º£º£º
1) 53ݪֲÎᆱÓÍɱÓ׳æ»îÐÔµÄɸѡ¼°Æä¶ÔäåÇè¾Õõ¥¿¹°×ÎÆÒÁÎÃÔöЧ×÷ÓõÄÑо¿£¬½ÃÅÊÐ2019-2020Äê¶È×ÔÈ»¿ÆÑ§ÓÅÒìѧÊõÂÛÎÄ£¬¶þµÈ½±£¬ÅÅÃûµÚÒ»£¬½ÃÅÊпÆÑ§ÊÖÒÕлᣬ2021Äê10Ô¡£¡£¡£
2) ѧУ¡¢¡¢ÐÐÒµÉî¶ÈÈںϡ°3+1¡±Ä£Ê½ÐͬÓýÈËÁ¢ÒìÓëʵ¼ù£¬Ò¼ºÅÓéÀÖAPPµÚÊ®Îå´Î½ÌѧЧ¹û½±£¬¶þµÈ½±£¬ÅÅÃûµÚËÄ£¬Ò¼ºÅÓéÀÖAPP£¬2019Äê5Ô¡£¡£¡£
3) Èâ¹ðËáõ¥ÀàÑÜÉúÎï×÷ΪÀÒ°±ËáøÒÖÖÆ¼ÁµÄÉè¼Æ¡¢¡¢ºÏ³É¼°ÆÀ¼Û£¬½ÃÅÊÐ2017-2018Äê¶È×ÔÈ»¿ÆÑ§ÓÅÒìѧÊõÂÛÎÄ£¬ÈýµÈ½±£¬ÅÅÃûµÚÒ»£¬½ÃÅÊпÆÑ§ÊÖÒÕлᣬ2019Äê9Ô¡£¡£¡£